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| Item No | Product Name | Product Description | Product Description | Inquiry |
|---|---|---|---|---|
| R-SX-444 | Dronedarone Hydrochloride,CAS141625-93-6 | Dronedarone HCl is a therapy for the treatment of patients with paroxysmal and persistent atrial fibrillation or atrial flutter.西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-445 | Fasudil; HA-1077,CAS203911-27-7 | HA-1077 inhibits vascular smooth muscle contraction by acting as an intracellular Ca2+ antagonist.西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-446 | PTC124,CAS775304-57-9 | Ataluren (PTC124) selectively induces ribosomal read-through of premature but not normal termination codons, with EC50 of 0.1 μM in HEK293 cells, may provide treatment for genetic disorders caused by nonsense mutations (e.g. CF caused by CFTR nonsense mutation). Phase 3.西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-447 | Vinpocetine,CAS42971-09-5 | Vinpocetine is a selective inhibitor of voltage-sensitive sodium channel for the treatment of stroke, vascular dementia and Alzheimer's disease.西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-448 | CB-5083,CAS1542705-92-9 | CB-5083是有效，选择性和有口服活性的 p97 抑制剂，IC50 值为 11 nM。西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-449 | LCZ696;Sacubitril;Valsartan，CAS172732-68-2 | Varespladib (LY315920) 是一种有效且具有选择性的 group IIA, secretory phospholipase A2 (sPLA2) 抑制剂，其 IC50 值为 9 nM。Varespladib 对大鼠，兔，豚鼠和人等各种物种血清的 sPLA2 活性具有明显的抑制作用，IC50 分别为 8.1 nM，5.0 nM，3.2 nM 和 6.2 nM。 西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-450 | Abiraterone Acetate; CB7630,CAS154229-18-2 | Abiraterone acetate 是一种口服、有效、选择性和不可逆的 CYP17A1 抑制剂，具有抗雄激素活性。Abiraterone acetate是 Abiraterone (CB7598) 的前药形式。 西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-451 | Abiraterone; CB7598,CAS154229-19-3 | Abiraterone is a potent CYP17 inhibitor with IC50 of 2 nM in a cell-free assay.西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-452 | Bexarotene,CAS153559-49-0 | Bexarotene is a retinoid specifically selective for retinoid X receptors, used as an oral antineoplastic agent in the treatment of cutaneous T-cell lymphoma.西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-453 | TOK001; VN1241，CAS851983-85-2 | Galeterone is a selective CYP17 inhibitor and androgen receptor (AR) antagonist with IC50 of 300 nM and 384 nM, respectively, and is a potent inhibitor of human prostate tumor growth. Phase 2.西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-454 | Anacetrapib; MK0859,CAS875446-37-0 | Anacetrapib 是一种有效的 CETP 抑制剂，作用于 rhCETP 和 C13S CETP 突变型，IC50 分别为 7.9±2.5 nM 和 11.8±1.9 nM。 西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-455 | Apremilast; CC10004,CAS608141-41-9 | Apremilast (CC-10004) is a potent and orally active PDE4 and TNF-α inhibitor with IC50 of 74 nM and 77 nM, respectively.西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
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