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| Item No | Product Name | Product Description | Product Description | Inquiry |
|---|---|---|---|---|
| R-SX-383 | MPEP hydrochloride,CAS219911-35-0 | MPEP is a potent, highly selective non-competitive antagonist at the mGlu5a receptor subtype (IC50 = 36 nM) while having no agonist or antagonist activities at the mGlu1b receptor at concentrations up to 30 uM.西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-384 | TG6-10-1,CAS1415716-58-3 | TG6-10-1 是一种 EP2 拮抗剂, 低纳摩尔下有效作用于 EP2, 比作用于人 EP3, EP4 和 IP 受体选择性高 300, EP1 受体选择性高 100 倍的。西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-385 | Elacridar HCl,CAS143851-98-3 | Elacridar hydrochloride is a P-glycoprotein inhibitor, and has been used both in vitro and in vivo as a tool inhibitor of P-glycoprotein (Pgp) to investigate the role of transporters in the disposition of various test molecules.西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-386 | Muscimol HBr,CAS18174-72-6 | Muscimol hydrobromide is a potent but toxic structural analog of g-aminobutyric acid (GABA), with a zwitterionic structure西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-388 | MK-801 ; Dizocilpine,CAS77086-21-6 | MK-801 (Dizocilpine) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM.西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-389 | Iloperidone,CAS133454-47-4 | Iloperidone(HP 873)是D2/5-HT2受体拮抗剂，可作用于精神分裂症。西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-390 | Bromfenac sodium,CAS91714-93-1 | Bromfenac Sodium是一种非甾体类抗炎药(NSAID)，具有抗炎活性，通过抑制环氧合酶1和2可阻断前列腺素的合成。西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-391 | VU0361737,CAS1161205-04-4 | VU 0361737 is a selective positive allosteric modulator (PAM) for mGlu4 receptor with EC50 of 240 nM and 110 nM at human and rat receptors, respectively, displays weak activity at mGlu5 and mGlu8 receptors, is inactive at mGlu1, mGlu2, mGlu3, mGlu6 and mGlu7 receptors, can penetrate into CNS.西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-392 | VU0357121,CAS433967-28-3 | VU0357121 is a novel positive allosteric modulator (PAM) of mGlu5 with EC50 of 33 nM, is inactive or very weakly antagonizing at other mGlu receptor subtypes.西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-393 | VU0364770,CAS61350-00-3 | VU 0364770 is a positive allosteric modulator(PAM) of mGlu4 with EC50 of 1.1 μM, exhibits insignificant activity at 68 other receptors, including other mGlu subtypes.西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-394 | Ivabradine hydrochloride,CAS148849-67-6 | Ivabradine hydrochloride 是可口服的，超极化激活的环核苷酸门控离子通道 (HCN) 通道阻滞剂。西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
| R-SX-395 | BRL54443,CAS57477-39-1 | BRL 54443是5-HT1E/1F受体激动剂，pKi分别为8.7和8.9，比对其它5-HT和多巴胺受体的抑制性高30倍以上。西安瑞禧生物提供各种抑制剂材料。 | 查看详细 | |
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